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An Expedient Synthesis of CMF-019: (S)-5-Methyl-3-{1-(pentan-3-yl)-2-(thiophen-2-ylmethyl)-1H-benzo[d]imidazole-5-carboxamido}hexanoic acid, an Apelin Receptor (APJ) Agonist.

Trifonov L.; Afri M.; Palczewski K.; Korshin E*. and Gruzman A*., 2018

Medicinal Chemistry, 2018, 14: 688 – 694.